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§ Encyclopedia · STRONG (A)
A

Strong

≥2 well-powered RCTs in humans with consistent effect size. Plausible mechanism. No major contradictory data.

# Compound Category EU Status Last reviewed
001. Bremelanotide
INN · bremelanotidum
Melanocortin (MC1R/MC3R/MC4R) receptor agonist · on-demand subcutaneous
Hormonal NOT AUTHORISED 18 MAY 2026
002. Setmelanotide
INN · setmelanotidum
MC4R-selective melanocortin receptor agonist · daily subcutaneous
Hormonal AUTHORISED 18 MAY 2026
003. Tesamorelin
INN · tesamorelinum
Synthetic GHRH analogue · stimulates pituitary GH release · daily subcutaneous
Metabolic AUTHORISED 18 MAY 2026